Palladium-catalyzed direct arylation of heteroarenes with aryl mesylates

Chau Ming So; Chak Po Lau; Fuk Yee Kwong

doi:10.1002/chem.201002354

Palladium-catalyzed direct arylation of heteroarenes with aryl mesylates

Chau Ming So, Chak Po Lau, Fuk Yee Kwong

Research output: Journal article publication › Journal article › Academic research › peer-review

91 Citations (Scopus)

Abstract

Not so challenging after all! The first general examples of the direct arylation of heteroarenes by using challenging aryl mesylates as electrophiles are disclosed. These easy reaction conditions also allow the functionalization of other heterocycles, such as caffeine, triazole and benzathiazole (see scheme).

Original language	English
Pages (from-to)	761-765
Number of pages	5
Journal	Chemistry - A European Journal
Volume	17
Issue number	3
DOIs	https://doi.org/10.1002/chem.201002354
Publication status	Published - 17 Jan 2011

Keywords

aryl mesylates
C-H activation
direct arylation
heterocycles
palladium

ASJC Scopus subject areas

General Chemistry

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10.1002/chem.201002354

Cite this

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title = "Palladium-catalyzed direct arylation of heteroarenes with aryl mesylates",

abstract = "Not so challenging after all! The first general examples of the direct arylation of heteroarenes by using challenging aryl mesylates as electrophiles are disclosed. These easy reaction conditions also allow the functionalization of other heterocycles, such as caffeine, triazole and benzathiazole (see scheme).",

keywords = "aryl mesylates, C-H activation, direct arylation, heterocycles, palladium",

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year = "2011",

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AB - Not so challenging after all! The first general examples of the direct arylation of heteroarenes by using challenging aryl mesylates as electrophiles are disclosed. These easy reaction conditions also allow the functionalization of other heterocycles, such as caffeine, triazole and benzathiazole (see scheme).

KW - aryl mesylates

KW - C-H activation

KW - direct arylation

KW - heterocycles

KW - palladium

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Palladium-catalyzed direct arylation of heteroarenes with aryl mesylates

Abstract

Keywords

ASJC Scopus subject areas

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